| 任学状,李雁武,郭卿,袁勇,袁建勇.化学通报,2015,78(12):1108-1112. |
| 醋酸特拉司酮的合成 |
| Synthesis of telapristone acetate |
| 投稿时间：2015-05-07 修订日期：2015-07-04 |
| DOI： |
| 中文关键词: 醋酸特拉司酮 醋酸乌利司他 合成 |
| 英文关键词:Telapristone acetate Uliprista Synthesis”应改为“Telapristone acetate Uliprista acetate Synthesis |
| 基金项目:重庆市教委技术研究项目（KJZH14204）资助 |
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| 中文摘要: |
| 以醋酸乌利司他为起始原料，乙二醇选择性保护3-羰基得到缩酮物，然后经21-甲基碘代、取代、水解、甲基化，最后脱保护，酯化得到醋酸特拉司酮。 |
| 英文摘要: |
| Telapristone acetate was synthesized from ulipristal acetate as the starting material through protection of the 3-Carbonyl group, iodination, substitution, methylation, deprotection of 3-carbonyl and acetylation of 17-hydroxy group. |
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